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St. John's Wort Drug Interactions

This content is for informational purposes only and does not constitute medical advice. Statements about dietary supplements have not been evaluated by the FDA and are not intended to diagnose, treat, cure, or prevent any disease. Individual results may vary — consult your healthcare provider before starting any supplement. Full disclaimer

St.

St. John's wort, sold over the counter for mood, is one of the most potent drug-interacting supplements known. It speeds up the breakdown of many medicines — weakening birth control, some heart, HIV, cancer, and transplant drugs — and can raise serotonin-syndrome risk with antidepressants. Don't combine it with medications without medical guidance.

Key Takeaways

  • St. John's wort speeds up drug-metabolizing enzymes, lowering levels of many medicines.
  • It can weaken birth control, heart, HIV, cancer, and transplant (cyclosporine) medications.
  • Combined with antidepressants or other serotonergic drugs, it can raise serotonin-syndrome risk.
  • Because it's an over-the-counter mood product, it's often left off medication lists.
  • Don't combine it with prescription medicines without medical guidance, and don't start or stop abruptly.

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A plant with a drug-like interaction profile

Despite being sold over the counter for low mood, St. John's wort has an interaction profile rivaling many prescription drugs. NCCIH states plainly that 'interactions with St. John's wort can weaken the effects of life-saving medicines or cause dangerous side effects' [1].

How it weakens medicines

St. John's wort induces (speeds up) drug-metabolizing enzymes, so the body clears affected medicines faster, lowering their blood levels and effectiveness [1]. NCCIH lists examples it can weaken [1]:

  • Birth control pills (risk of unintended pregnancy) — see [supplements and birth control](/learn/supplements-and-birth-control)
  • Heart medicines such as digoxin and ivabradine
  • HIV medicines such as indinavir and nevirapine
  • Cancer medicines such as irinotecan, imatinib, and docetaxel
  • Transplant anti-rejection medicines such as cyclosporine — see [supplements and immunosuppressants](/learn/supplements-and-immunosuppressants)

The serotonin risk

Separately, St. John's wort raises serotonin activity, so combining it 'with certain antidepressants or other drugs that affect serotonin...may lead to increased serotonin-related side effects, which can be serious' [1] — see serotonin syndrome and supplements.

Why it's so often missed

Because it's a herbal product for mood, people don't list it as a medication — yet weakening a transplant or HIV drug can have severe consequences. The stakes make disclosure essential [2].

Practical guidance

  • Tell every provider and pharmacist if you take or are considering St. John's wort.
  • Don't combine it with prescription medicines without medical clearance, especially the categories above.
  • Don't start or stop it abruptly around a medication change — stopping it can raise the level of a drug it was speeding up.
  • Treat it with the same seriousness as a prescription drug when reviewing interactions.

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Frequently Asked Questions

Why is St. John's wort such a problem with medications?

It induces, or speeds up, the enzymes that break down many drugs, so it lowers their blood levels and can make them less effective. NCCIH warns it can weaken life-saving medicines, and it also raises serotonin activity, adding a separate risk with antidepressants.

Which medications does St. John's wort affect?

NCCIH lists birth control pills, heart medicines like digoxin and ivabradine, HIV drugs like indinavir and nevirapine, cancer drugs like irinotecan and imatinib, and transplant anti-rejection medicines like cyclosporine, among others. Its interaction list is unusually broad.

Can I take St. John's wort if I'm on antidepressants?

Not without medical guidance. Combining St. John's wort with antidepressants or other serotonin-affecting drugs can lead to serious serotonin-related side effects. If you take an antidepressant, talk to your prescriber before considering St. John's wort.

Is it safe to stop St. John's wort suddenly?

Stopping it changes drug metabolism, which can raise the level of a medicine it was speeding up — so abrupt changes around other medications should be managed with a clinician. The broader point is to involve your provider whenever St. John's wort and prescription drugs overlap.

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References

  1. National Center for Complementary and Integrative Health (2025). St. John's Wort: Usefulness and Safety. U.S. National Institutes of Health.
  2. National Center for Complementary and Integrative Health (2026). How Medications and Supplements Can Interact. U.S. National Institutes of Health.